SCHEMBL8235332

SCHEMBL8235332

C[C@H](N)C(=O)NC(=N)c1ccc(N2CCN(c3nc(-c4ccncn4)cc(=O)n3C)[C@H](C)C2)cc1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 20/20 0.67
CYP2D6 P10635 10/20 0.66
CYP1A2 P05177 8/20 0.66
CYP3A4 P08684 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8231884 0.90 GSK3B (0.55) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL698204 0.88 GSK3B (0.76) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL8232490 0.87 GSK3B (0.67) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL8232515 0.85 GSK3B (0.68) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL697457 0.84 GSK3B (0.81) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL8227140 0.84 GSK3B (0.63) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL697339 0.82 GSK3B (0.85) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL697856 0.81 GSK3B (1.00) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL13712789 0.81 GSK3B (0.76) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL13711549 0.81 GSK3B (0.76) GSK3BCYP2D6CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007119463-A1 2-(CYCLIC AMINO)-PYRIMIDONE DERIVATIVES AS TPK1 INHIBITORS MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-10-25 WO disclosed