SCHEMBL8238773

SCHEMBL8238773

CC(C)(C)OC(=O)N1CCNC[C@H]1Cc1ccc(C(=O)O)cc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.54
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA4 P22748 2/20 0.48
CA9 Q16790 2/20 0.48
NR1H2 P55055 2/20 0.45
NR1H3 Q13133 2/20 0.45
HDAC1 Q13547 1/20 0.43
DPP4 P27487 5/20 0.40
REN P00797 2/20 0.40
DPP7 Q9UHL4 2/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL873458 0.90 PARP1 (0.54) PARP1CA1CA2CA4CA9
SCHEMBL4309187 0.90 PARP1 (0.54) PARP1CA1CA2CA4CA9
SCHEMBL873429 0.90 PARP1 (0.54) PARP1CA1CA2CA4CA9
SCHEMBL874327 0.88 PARP1 (0.56) PARP1CA1CA2CA4CA9
SCHEMBL15205855 0.88 PARP1 (0.56) PARP1CA1CA2CA4CA9
SCHEMBL5359873 0.87 PARP1 (0.55) PARP1CA1CA2CA4CA9
SCHEMBL27933734 0.87 PARP1 (0.55) PARP1CA1CA2CA4CA9
SCHEMBL873810 0.87 PARP1 (0.55) PARP1CA1CA2CA4CA9
SCHEMBL874539 0.86 PARP1 (0.54) PARP1CA1CA2CA4CA9
SCHEMBL5365387 0.85 PARP1 (0.53) PARP1CA1CA2CA4CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007094513-A2 CYCLIC AMINE COMPOUND AND USE THEREOF FOR THE PROPHYLAXIS OR TREATMENT OF HYPERTENSION TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-08-23 WO disclosed