SCHEMBL8239282

SCHEMBL8239282

Cc1cc(F)ccc1-c1cc(N2CCN3CCCC3C2=O)ncc1N(C)C(=O)C1(c2cc(C(F)(F)F)cc(C(F)(F)F)c2)CC1

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 18/20 0.52
TACR3 P29371 9/20 0.52
CYP3A4 P08684 10/20 0.50
GPBAR1 Q8TDU6 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8239455 1.00 TACR1 (0.52) TACR1TACR3CYP3A4GPBAR1
SCHEMBL10182983 1.00 TACR1 (0.52) TACR1TACR3CYP3A4GPBAR1
SCHEMBL8251136 0.90 TACR1 (0.51) TACR1TACR3CYP3A4
SCHEMBL10181750 0.89 TACR1 (0.51) TACR1TACR3CYP3A4GPBAR1
SCHEMBL337288 0.87 TACR1 (0.68) TACR1TACR3CYP3A4
SCHEMBL10182959 0.87 TACR1 (0.68) TACR1TACR3CYP3A4
SCHEMBL12583015 0.86 TACR1 (0.51) TACR1TACR3CYP3A4GPBAR1
SCHEMBL337076 0.85 TACR1 (0.58) TACR1TACR3CYP3A4GPBAR1
SCHEMBL337573 0.85 TACR1 (0.58) TACR1TACR3CYP3A4GPBAR1
SCHEMBL12582965 0.85 TACR1 (0.58) TACR1TACR3CYP3A4GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007028654-A1 PYRIDINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF PSYCHOTIC DISORDERS SMITHKLINE BEECHAM CORPORATION (US) 2007-03-15 WO disclosed