SCHEMBL8245646

SCHEMBL8245646

O=C(O)CNC(=O)c1c(O)c2cc(C(F)(F)F)ccc2n(Cc2ccccc2Cl)c1=O

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGLN3 Q9H6Z9 6/20 0.69
EGLN1 Q9GZT9 10/20 0.64
EGLN2 Q96KS0 4/20 0.64
CYSLTR2 Q9NS75 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
NPC1 O15118 1/20 0.47
HIF1A Q16665 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8244838 0.93 EGLN3 (0.78) EGLN3EGLN1EGLN2CYSLTR2MEN1
SCHEMBL8247226 0.88 EGLN3 (0.85) EGLN3EGLN1EGLN2MEN1KMT2A
SCHEMBL5311749 0.88 EGLN3 (0.72) EGLN3EGLN1EGLN2MEN1KMT2A
SCHEMBL5309011 0.84 EGLN1 (0.73) EGLN3EGLN1EGLN2CYSLTR2HIF1A
SCHEMBL8238784 0.83 EGLN3 (0.67) EGLN3EGLN1EGLN2MEN1KMT2A
SCHEMBL8248296 0.82 EGLN3 (1.00) EGLN3EGLN1EGLN2MEN1KMT2A
SCHEMBL8244813 0.82 EGLN1 (0.57) EGLN3EGLN1EGLN2CYSLTR2HIF1A
SCHEMBL8248494 0.81 EGLN1 (0.75) EGLN3EGLN1EGLN2CYSLTR2HIF1A
SCHEMBL8247380 0.81 EGLN3 (0.74) EGLN3EGLN1EGLN2HIF1A
SCHEMBL8247316 0.81 EGLN3 (0.74) EGLN3EGLN1EGLN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007038571-A2 PROLYL HYDROXYLASE ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2007-04-05 WO disclosed