SCHEMBL8247787

SCHEMBL8247787

CCCOCCn1c(=O)c(NCCNC)nc2cnc(-c3ccc(OC)nc3)cc21

nearest known ligand 0.84

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 20/20 0.84
PDE6A P16499 20/20 0.84
KCNH2 Q12809 1/20 0.82
PDE11A Q9HCR9 2/20 0.76
PDE4B Q07343 1/20 0.70
PDE4D Q08499 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8250277 0.92 PDE5A (0.86) PDE5APDE6AKCNH2PDE11APDE4B
SCHEMBL5813631 0.92 PDE5A (0.89) PDE5APDE6AKCNH2PDE11APDE4B
SCHEMBL8248115 0.92 PDE5A (0.91) PDE5APDE6AKCNH2PDE11APDE4B
SCHEMBL5814292 0.92 PDE5A (1.00) PDE5APDE6AKCNH2PDE11A
SCHEMBL8240941 0.92 PDE5A (1.00) PDE5APDE6AKCNH2PDE11APDE4B
SCHEMBL5820167 0.92 PDE5A (1.00) PDE5APDE6AKCNH2PDE11APDE4B
SCHEMBL8247767 0.91 PDE5A (0.81) PDE5APDE6AKCNH2PDE11A
SCHEMBL5813844 0.90 PDE5A (0.82) PDE5APDE6AKCNH2PDE11A
SCHEMBL5812288 0.90 PDE5A (1.00) PDE5APDE6AKCNH2PDE11A
SCHEMBL8250774 0.90 PDE5A (1.00) PDE5APDE6AKCNH2PDE11APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006126083-A1 PYRIDINE [3 , 4-B] PYRAZINONE COMPOUNDS AS PDE-5 INHIBITORS PHARMACIA & UPJOHN COMPANY LLC (US) 2006-11-30 WO disclosed