SCHEMBL8248262

SCHEMBL8248262

CC(=O)NC(=O)C(I)C(C)C

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 1/20 0.38
TAS2R38 P59533 1/20 0.35
KDM4E B2RXH2 1/20 0.32
CA2 P00918 1/20 0.32
PTGS1 P23219 1/20 0.32
MMP12 P39900 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ALPL P05186 1/20 0.32
APOBEC3G Q9HC16 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
NFKB1 P19838 1/20 0.30
EPHX1 P07099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11458390 0.77
SCHEMBL10575445 0.77 CRBN (0.42) CRBNCA2ALDH1A1NFKB1
SCHEMBL12435336 0.76 CRBN (0.39) CRBNTAS2R38KDM4ECA2PTGS1
SCHEMBL12512722 0.76 CRBN (0.39) CRBNTAS2R38KDM4ECA2PTGS1
SCHEMBL2220319 0.75
SCHEMBL10942414 0.75 CRBN (0.43) CRBNTAS2R38KDM4ECA2PTGS1
SCHEMBL6517566 0.72
SCHEMBL29616779 0.72 DPP4 (0.48) CRBNTAS2R38KDM4ECA2PTGS1
SCHEMBL25458289 0.70
SCHEMBL29616787 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007002173-A1 HIV-1 PROTEASE INHIBITORS, AND METHODS OF MAKING AND USING THEM UNIVERSITY OF MASSACHUSETTS (US) 2007-01-04 WO disclosed