SCHEMBL8248993

SCHEMBL8248993

C[C@@H]1C[C@@H](C(=O)N[C@@H](CNC(=O)NCc2ccccc2)C(=O)O)N(S(=O)(=O)c2ccccc2)C1

nearest known ligand 0.70

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 13/20 0.70
ITGA2 P17301 7/20 0.70
ITGA4 P13612 2/20 0.63
FKBP1A P62942 1/20 0.43
CAPN1 P07384 2/20 0.42
CTSB P07858 1/20 0.42
ITGAV P06756 3/20 0.42
ALDH1A1 P00352 2/20 0.42
ITGA5 P08648 3/20 0.42
USP2 O75604 1/20 0.41
ITGB3 P05106 1/20 0.41
MMP1 P03956 1/20 0.41
MMP3 P08254 1/20 0.41
MMP7 P09237 1/20 0.41
MMP9 P14780 1/20 0.41
MMP13 P45452 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4249877 0.92 ITGB1 (0.71) ITGB1ITGA2ITGA4FKBP1ACAPN1
SCHEMBL12084795 0.92 ITGB1 (0.71) ITGB1ITGA2ITGA4FKBP1ACAPN1
SCHEMBL4259018 0.86 ITGB1 (0.66) ITGB1ITGA2ITGA4FKBP1ACAPN1
SCHEMBL8245234 0.86 ITGB1 (0.66) ITGB1ITGA2ITGA4FKBP1ACAPN1
SCHEMBL1487410 0.85 ITGB1 (0.75) ITGB1ITGA2ITGA4FKBP1AITGAV
SCHEMBL8239058 0.84 ITGB1 (0.83) ITGB1ITGA2ITGA4FKBP1AITGAV
SCHEMBL12084502 0.84 ITGB1 (0.83) ITGB1ITGA2ITGA4FKBP1AITGAV
SCHEMBL4255594 0.84 ITGB1 (0.83) ITGB1ITGA2ITGA4FKBP1AITGAV
SCHEMBL12084791 0.83 ITGB1 (0.79) ITGB1ITGA2ITGA4FKBP1AITGAV
SCHEMBL4260019 0.83 ITGB1 (0.79) ITGB1ITGA2ITGA4FKBP1AITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006133338-A1 INHIBITORS OF THE α2β1/GPIa-IIa INTEGRIN THE TRUSTEES OF THE UNIVERSITY OF PENNESYLVANIA (US) 2006-12-14 WO disclosed