SCHEMBL8249103

SCHEMBL8249103

C=C(O)[C@H](CNC(=O)NCc1ccc(-c2ccccc2)cc1)NC(=O)[C@@H]1CCCN1S(=O)(=O)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 7/20 0.59
ITGA2 P17301 4/20 0.59
ITGA4 P13612 1/20 0.59
MMP2 P08253 3/20 0.50
MMP9 P14780 2/20 0.50
FKBP1A P62942 4/20 0.49
ITGA5 P08648 2/20 0.45
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
ITGAV P06756 1/20 0.43
SCN9A Q15858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4253387 0.94 ITGB1 (0.68) ITGB1ITGA2ITGA4MMP2MMP9
SCHEMBL12084495 0.94 ITGB1 (0.68) ITGB1ITGA2ITGA4MMP2MMP9
SCHEMBL8244929 0.92 ITGB1 (0.55) ITGB1ITGA2ITGA4MMP2MMP9
SCHEMBL8238713 0.92 ITGB1 (0.69) ITGB1ITGA2ITGA4MMP2MMP9
SCHEMBL4251535 0.90 ITGB1 (0.73) ITGB1ITGA2ITGA4MMP2MMP9
SCHEMBL8245510 0.90 ITGB1 (0.73) ITGB1ITGA2ITGA4MMP2MMP9
SCHEMBL8248434 0.88 ITGB1 (0.72) ITGB1ITGA2ITGA4MMP2MMP9
SCHEMBL8245644 0.87 ITGB1 (0.64) ITGB1ITGA2ITGA4MMP2MMP9
SCHEMBL8248234 0.86 ITGB1 (0.65) ITGB1ITGA2ITGA4MMP2MMP9
SCHEMBL4260308 0.86 ITGB1 (0.65) ITGB1ITGA2ITGA4MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006133338-A1 INHIBITORS OF THE α2β1/GPIa-IIa INTEGRIN THE TRUSTEES OF THE UNIVERSITY OF PENNESYLVANIA (US) 2006-12-14 WO disclosed