SCHEMBL8249691

SCHEMBL8249691

CCC1(c2ccccc2C)CCN(C(=O)c2cn(Cc3cccnc3)c3cc(Cl)ccc23)CC1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 8/20 0.46
CNR1 P21554 2/20 0.44
CNR2 P34972 1/20 0.44
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP46A1 Q9Y6A2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CHRM2 P08172 1/20 0.38
ADRA1D P25100 1/20 0.38
TACR3 P29371 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8251835 0.86 AVPR1A (0.48) AVPR1ACNR1MEN1KMT2AADRA1D
SCHEMBL4361153 0.82 AVPR1A (0.57) AVPR1ACNR1CNR2MEN1KMT2A
SCHEMBL8241424 0.81 AVPR1A (0.69) AVPR1ACNR1ALDH1A1
SCHEMBL4359158 0.81 AVPR1A (0.69) AVPR1ACNR1CNR2MEN1KMT2A
SCHEMBL4359118 0.81 AVPR1A (0.55) AVPR1ACNR1CNR2MEN1KMT2A
SCHEMBL8251337 0.79 AVPR1A (0.51) AVPR1ACNR1ALDH1A1
SCHEMBL8249649 0.78 AVPR1A (0.50) AVPR1ACNR1ALDH1A1
SCHEMBL13971309 0.77 AVPR1A (0.44) AVPR1ACNR1KMT2AALDH1A1
SCHEMBL14580413 0.76 AVPR1A (0.46) AVPR1ACNR1CNR2MEN1KMT2A
SCHEMBL613261 0.74 CNR1 (0.43) CNR1CNR2MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007006688-A1 INDOL-3-CARBONYL-SPIRO-PIPERIDINE DERIVATIVES AS V1A RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2007-01-18 WO disclosed