SCHEMBL8250210

SCHEMBL8250210

C#Cc1ccc(CN2CCN(Cc3cc(Cl)c4c(c3)CN(Cc3ccc(OC(F)(F)F)cc3)C4=O)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
GRM2 Q14416 2/20 0.45
TSHR P16473 1/20 0.44
LSS P48449 1/20 0.38
KCNH2 Q12809 1/20 0.37
DRD4 P21917 2/20 0.36
DRD2 P14416 1/20 0.36
CHRM5 P08912 1/20 0.36
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
BACE1 P56817 1/20 0.36
HCRTR1 O43613 2/20 0.36
HCRTR2 O43614 2/20 0.36
GRIN2B Q13224 2/20 0.36
PRCP P42785 1/20 0.35
ABL1 P00519 1/20 0.35
GPR6 P46095 1/20 0.35
TNF P01375 1/20 0.35
NOD2 Q9HC29 1/20 0.35
NOD1 Q9Y239 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12413538 0.91 GRM2 (0.47) ALDH1A1GRM2TSHRLSSKCNH2
SCHEMBL2022539 0.87 GRM2 (0.44) ALDH1A1GRM2TSHRCHRM5HCRTR1
SCHEMBL2024727 0.84 GRM2 (0.44) ALDH1A1GRM2TSHRDRD4GPR6
SCHEMBL12580818 0.83 GPR6 (0.46) ALDH1A1GRM2TSHRKCNH2GPR6
SCHEMBL2026888 0.82 GRM2 (0.47) ALDH1A1GRM2TSHRCHRM5HCRTR1
SCHEMBL1001844 0.82 GRM2 (0.43) ALDH1A1GRM2TSHRBCHEACHE
SCHEMBL1001587 0.82 GRM2 (0.42) ALDH1A1GRM2TSHRKCNH2CHRM5
SCHEMBL2022149 0.81 HTT (0.48) ALDH1A1GRM2TSHRDRD4DRD2
SCHEMBL8246819 0.81 GRM2 (0.45) ALDH1A1GRM2TSHRCHRM5HCRTR1
SCHEMBL2026639 0.81 GRM2 (0.47) ALDH1A1GRM2TSHRCHRM5HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007021309-A1 SUBSTITUTED ISOINDOLONES AND THEIR USE AS METABOTROPIC GLUTAMATE RECEPTOR POTENTIATORS ASTRAZENECA AB (SE) 2007-02-22 WO disclosed