SCHEMBL8251392

SCHEMBL8251392

CCC(C)n1c(=O)n(CC)c(=O)c2[nH]c(C34CC5CC(CC3C5)C4)nc21

nearest known ligand 0.75

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.64
ADORA2B P29275 9/20 0.64
ADORA1 P30542 7/20 0.64
ADORA3 P0DMS8 5/20 0.64
SLC6A3 Q01959 1/20 0.64
SLC22A6 Q4U2R8 1/20 0.64
SLC22A8 Q8TCC7 1/20 0.64
SLC22A11 Q9NSA0 1/20 0.64
MEN1 O00255 1/20 0.57
MAPT P10636 1/20 0.57
KMT2A Q03164 1/20 0.57
SIRT2 Q8IXJ6 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
SIRT3 Q9NTG7 1/20 0.36
SIRT5 Q9NXA8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7269103 0.86 ADORA1 (0.81) ADORA2AADORA2BADORA1ADORA3SLC6A3
SCHEMBL14051422 0.83 ADORA1 (0.91) ADORA2AADORA2BADORA1ADORA3SLC6A3
Rolofylline SCHEMBL720438 0.78 ADORA1 (1.00) ADORA2AADORA2BADORA1ADORA3SLC6A3
SCHEMBL7270718 0.77 ADORA1 (1.00) ADORA2AADORA2BADORA1ADORA3SLC6A3
SCHEMBL8704620 0.76 ADORA1 (0.81) ADORA2AADORA2BADORA1ADORA3SLC6A3
Rolofylline SCHEMBL13414143 0.76 ADORA1 (0.78) ADORA2AADORA2BADORA1ADORA3SLC6A3
SCHEMBL8709754 0.75 ADORA1 (0.83) ADORA2AADORA2BADORA1ADORA3SLC6A3
SCHEMBL7279878 0.75 ADORA1 (0.72) ADORA2AADORA2BADORA1ADORA3SLC6A3
Rolofylline SCHEMBL13414105 0.74 ADORA1 (0.86) ADORA2AADORA2BADORA1ADORA3SLC6A3
SCHEMBL7270716 0.74 ADORA1 (0.82) ADORA2AADORA2BADORA1ADORA3SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006115690-A2 PRODUCTION OF EMULSIONS FOR INTRAVENOUS INJECTION OF WATER-INSOLUBLE PHARMACEUTICAL COMPOSITIONS NOVACARDIA, INC. (US) 2006-11-02 WO disclosed