SCHEMBL8257828

SCHEMBL8257828

CC(C)C[C@H](NC(=O)[C@@H](NC(=O)c1ccc(-c2ccccc2)cn1)C(C)O)B(O)O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 15/20 0.68
PSMB1 P20618 6/20 0.68
PSMB8 P28062 6/20 0.68
PSMB9 P28065 6/20 0.68
PSMB10 P40306 6/20 0.68
PSMB2 P49721 6/20 0.68
ELANE P08246 2/20 0.68
CTSG P08311 2/20 0.68
CMA1 P23946 2/20 0.68
CYP3A4 P08684 1/20 0.68
LONP1 P36776 8/20 0.54
PSMB11 A5LHX3 5/20 0.54
PSMA7 O14818 5/20 0.54
PSMA1 P25786 5/20 0.54
PSMA2 P25787 5/20 0.54
PSMA3 P25788 5/20 0.54
PSMA4 P25789 5/20 0.54
PSMA5 P28066 5/20 0.54
PSMB4 P28070 5/20 0.54
PSMB6 P28072 5/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2934804 1.00 PSMB5 (0.68) PSMB5PSMB1PSMB8PSMB9PSMB10
SCHEMBL2934071 0.87 PSMB5 (0.73) PSMB5PSMB1PSMB8PSMB9PSMB10
SCHEMBL2936700 0.85 PSMB5 (0.68) PSMB5PSMB1PSMB8PSMB9PSMB10
SCHEMBL3164355 0.85 PSMB5 (0.67) PSMB5PSMB1PSMB8PSMB9PSMB10
SCHEMBL2927894 0.84 PSMB5 (0.70) PSMB5PSMB1PSMB8PSMB9PSMB10
SCHEMBL8259864 0.82 PSMB5 (0.64) PSMB5PSMB1PSMB8PSMB9PSMB10
SCHEMBL2933648 0.82 PSMB5 (0.64) PSMB5PSMB1PSMB8PSMB9PSMB10
SCHEMBL24195078 0.82 PSMB5 (0.78) PSMB5PSMB1PSMB8PSMB9PSMB10
SCHEMBL2933926 0.82 PSMB5 (0.78) PSMB5PSMB1PSMB8PSMB9PSMB10
SCHEMBL2930837 0.82 PSMB5 (0.72) PSMB5PSMB1PSMB8PSMB9PSMB10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006086600-A1 PROTEASOME INHIBITORS AND METHODS OF USING THE SAME CEPHALON, INC. (US) 2006-08-17 WO disclosed