SCHEMBL8258463

SCHEMBL8258463

COCC1=C(C(=O)OC(C)C)C(c2ccccc2I)C(C)=C(C)N1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 3/20 0.44
CYP1A2 P05177 4/20 0.41
CYP3A4 P08684 4/20 0.41
CYP2C9 P11712 4/20 0.41
CYP2C19 P33261 4/20 0.41
TBXA2R P21731 3/20 0.41
SLC6A3 Q01959 3/20 0.41
KCNH2 Q12809 3/20 0.41
CACNA1C Q13936 3/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
ALOX15 P16050 2/20 0.41
ABCB11 O95342 2/20 0.41
ADORA3 P0DMS8 2/20 0.41
OPRD1 P41143 2/20 0.41
OPRK1 P41145 2/20 0.41
SCN5A Q14524 2/20 0.41
CYP2D6 P10635 2/20 0.41
MLNR O43193 1/20 0.41
NR1I2 O75469 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8260790 0.89 NR3C2 (0.43) NR3C2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8260792 0.87 NR3C2 (0.42) NR3C2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL13587741 0.78 NR3C2 (0.58) NR3C2KDM4E
SCHEMBL13587768 0.76 NR3C2 (0.56) NR3C2KDM4E
SCHEMBL13587771 0.76 NR3C2 (0.56) NR3C2KDM4E
SCHEMBL13587767 0.76 NR3C2 (0.56) NR3C2TBXA2RSLC6A3KCNH2CACNA1C
SCHEMBL13587756 0.71 KDM4E (0.51) NR3C2TBXA2RALOX15ADORA3SCN5A
SCHEMBL8258936 0.71 NR3C2 (0.51) NR3C2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7431518 0.70 CACNA1C (0.53) NR3C2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8259167 0.70 KDM4E (0.54) NR3C2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006066011-A2 COMPOUNDS AND COMPOSITIONS AS MODULATORS OF STEROIDAL RECEPTORS AND CALCIUM CHANNEL ACTIVITIES IRM LLC (BM) 2006-06-22 WO disclosed