SCHEMBL8259100

SCHEMBL8259100

CS(=O)(=O)c1ccc2c(c1)nc1n2CC(N)[C@@H](c2cc(F)c(F)cc2F)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 1.00
DPP7 Q9UHL4 14/20 0.86
KCNH2 Q12809 5/20 0.86
CYP2D6 P10635 4/20 0.86
DPP9 Q86TI2 5/20 0.65
DPP8 Q6V1X1 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21067325 1.00 DPP4 (1.00) DPP4DPP7KCNH2CYP2D6DPP9
SCHEMBL8260956 0.92 DPP4 (0.86) DPP4DPP7KCNH2CYP2D6DPP9
SCHEMBL13342400 0.92 DPP4 (0.86) DPP4DPP7KCNH2CYP2D6DPP9
SCHEMBL13342409 0.85 DPP4 (0.87) DPP4DPP7KCNH2CYP2D6DPP9
SCHEMBL3535584 0.85 DPP4 (0.87) DPP4DPP7KCNH2CYP2D6DPP9
Trifluoroacetic Acid SCHEMBL3537790 0.85 DPP4 (1.00) DPP4DPP7KCNH2CYP2D6DPP9
SCHEMBL8261829 0.83 DPP4 (0.71) DPP4DPP7KCNH2CYP2D6DPP9
SCHEMBL2469613 0.83 DPP4 (0.71) DPP4DPP7KCNH2CYP2D6DPP9
SCHEMBL13342410 0.83 DPP4 (0.71) DPP4DPP7KCNH2CYP2D6DPP9
SCHEMBL13342393 0.80 DPP4 (0.82) DPP4DPP7KCNH2CYP2D6DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1819674-B1 FUSED AMINOPIPERIDINES AS DIPEPTIDYL PEPTIDASE-IV INHIBITORS FOR THE TREATMENT OR PREVENTION OF DIABETES MERCK SHARP & DOHME (US) 2011-10-05 EP disclosed
WO-2006058064-A2 FUSED AMINOPIPERIDINES AS DIPEPTIDYL PEPTIDASE-IV INHIBITORS FOR THE TREATMENT OR PREVENTION OF DIABETES MERCK & CO., INC. (US) 2006-06-01 WO disclosed