SCHEMBL8259153

SCHEMBL8259153

CC(CNCCCc1cccc(C(F)(F)F)c1)c1cccc2ccccc12

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.72
ADRA2C P18825 3/20 0.72
SLC6A4 P31645 3/20 0.72
DRD3 P35462 3/20 0.72
ADRB1 P08588 3/20 0.72
SLC6A2 P23975 2/20 0.72
OPRM1 P35372 2/20 0.72
CASR P41180 2/20 0.72
CYP2D6 P10635 2/20 0.72
HTT P42858 2/20 0.72
MLNR O43193 1/20 0.72
ABCB11 O95342 1/20 0.72
ADORA3 P0DMS8 1/20 0.72
CHRM1 P11229 1/20 0.72
DRD2 P14416 1/20 0.72
CHRM3 P20309 1/20 0.72
GLRA1 P23415 1/20 0.72
AVPR2 P30518 1/20 0.72
HRH1 P35367 1/20 0.72
MC3R P41968 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20307882 0.90 CASR (0.74) HTR2CADRA2CSLC6A4DRD3ADRB1
SCHEMBL23858339 0.85 CASR (0.73) HTR2CADRA2CSLC6A4DRD3ADRB1
SCHEMBL23858316 0.85 CASR (0.73) HTR2CADRA2CSLC6A4DRD3ADRB1
Cinacalcet SCHEMBL29360301 0.84 CASR (1.00) HTR2CADRA2CSLC6A4DRD3ADRB1
Cinacalcet SCHEMBL30371982 0.84 CASR (1.00) HTR2CADRA2CSLC6A4DRD3ADRB1
Cinacalcet SCHEMBL1901469 0.84 CASR (1.00) HTR2CADRA2CSLC6A4DRD3ADRB1
Cinacalcet SCHEMBL71876 0.84 CASR (1.00) HTR2CADRA2CSLC6A4DRD3ADRB1
Cinacalcet SCHEMBL29373418 0.84 CASR (1.00) HTR2CADRA2CSLC6A4DRD3ADRB1
Cinacalcet SCHEMBL3227084 0.84 CASR (1.00) HTR2CADRA2CSLC6A4DRD3ADRB1
SCHEMBL13855365 0.84 CASR (0.71) HTR2CADRA2CSLC6A4DRD3ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006125026-A2 PROCESS FOR PREPARING CINACALCET HYDROCHLORIDE TEVA PHARMACEUTICAL INDUSTRIES, LTD. (IL) 2006-11-23 WO disclosed