SCHEMBL8260705

SCHEMBL8260705

COC(=O)C1=C(C2CC2)NC(C)=C(C#N)C1c1ccc(F)cc1C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 2/20 0.50
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 3/20 0.41
ADORA3 P0DMS8 3/20 0.41
MAPT P10636 3/20 0.41
CYP2C9 P11712 3/20 0.41
CYP2C19 P33261 3/20 0.41
TSHR P16473 2/20 0.41
NFKB1 P19838 2/20 0.41
CACNA1C Q13936 2/20 0.41
MEN1 O00255 1/20 0.41
CYP2D6 P10635 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8260711 0.88 NR3C2 (0.62) NR3C2CYP1A2CYP3A4ADORA3MAPT
SCHEMBL8259588 0.87 NR3C2 (0.62) NR3C2MAPTTSHR
SCHEMBL13587784 0.86 NR3C2 (0.46) NR3C2CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL8260833 0.83 NR3C2 (0.47) NR3C2
SCHEMBL8261160 0.81 NR3C2 (0.50) NR3C2
SCHEMBL8259769 0.80 NR3C2 (0.48) NR3C2
SCHEMBL8259186 0.80 NR3C2 (0.49) NR3C2
SCHEMBL3812166 0.80 HTT (0.43) NR3C2CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL13587737 0.79 NR3C2 (0.49) NR3C2MAPTTSHRKMT2A
SCHEMBL8258517 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006066011-A2 COMPOUNDS AND COMPOSITIONS AS MODULATORS OF STEROIDAL RECEPTORS AND CALCIUM CHANNEL ACTIVITIES IRM LLC (BM) 2006-06-22 WO disclosed