SCHEMBL8264146

SCHEMBL8264146

Nc1ccccc1NC(=O)c1ccc(CNc2ncccc2CC(=O)C2CC2)cc1

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 19/20 0.65
HDAC3 O15379 7/20 0.54
HDAC2 Q92769 7/20 0.54
NCOR2 Q9Y618 5/20 0.54
HDAC8 Q9BY41 5/20 0.52
NCOR1 O75376 3/20 0.52
CYP3A4 P08684 1/20 0.52
HDAC11 Q96DB2 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1064336 0.81 HDAC1 (0.76) HDAC1HDAC3HDAC2NCOR2HDAC8
SCHEMBL1064069 0.80 HDAC1 (1.00) HDAC1HDAC3HDAC2NCOR2HDAC8
SCHEMBL1064400 0.76 HDAC1 (0.70) HDAC1HDAC3HDAC2NCOR2HDAC8
SCHEMBL1083540 0.72 HDAC1 (0.67) HDAC1HDAC3HDAC2NCOR2HDAC8
SCHEMBL210812 0.72 HDAC1 (0.79) HDAC1HDAC3HDAC2NCOR2HDAC8
SCHEMBL2414954 0.72 HDAC1 (0.69) HDAC1HDAC3HDAC2NCOR2HDAC8
SCHEMBL10814316 0.72 HDAC1 (0.59) HDAC1HDAC3HDAC2NCOR2HDAC8
SCHEMBL15518884 0.72 HDAC1 (1.00) HDAC1HDAC3HDAC2NCOR2HDAC8
SCHEMBL2413506 0.71 HDAC1 (0.68) HDAC1HDAC3HDAC2NCOR2HDAC8
SCHEMBL8348463 0.71 HDAC1 (0.83) HDAC1HDAC3HDAC2NCOR2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006066133-A2 HISTONE DEACETYLASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO disclosed