SCHEMBL8265124

SCHEMBL8265124

N=C/C=N\Nc1ccc(CN)cc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.37
LOXL2 Q9Y4K0 6/20 0.35
ABAT P80404 1/20 0.34
F10 P00742 1/20 0.34
F11 P03951 1/20 0.34
ST14 Q9Y5Y6 1/20 0.34
NOS3 P29474 2/20 0.32
NOS1 P29475 2/20 0.32
NOS2 P35228 2/20 0.32
TAAR1 Q96RJ0 1/20 0.32
TPSAB1 Q15661 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
NCOR2 Q9Y618 1/20 0.32
PLG P00747 1/20 0.31
PLAU P00749 1/20 0.31
PLAT P00750 1/20 0.31
KLKB1 P03952 1/20 0.31
PRSS1 P07477 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23969723 0.81 GRIN2D (0.38) HDAC3HDAC6PLAU
SCHEMBL22877058 0.75 GAA (0.47)
SCHEMBL20867958 0.74 HRH3 (0.44) HRH3LOXL2ABATF10F11
SCHEMBL18925387 0.69 MAPT (0.44) HDAC3HDAC6PLGPRSS1
SCHEMBL18059186 0.68 HRH3 (0.38) HRH3LOXL2ABATF10F11
SCHEMBL258907 0.65 HRH3 (0.55) HRH3LOXL2ABATF10F11
SCHEMBL27238704 0.64 HRH3 (0.79) HRH3LOXL2ABATF10F11
SCHEMBL15828 0.64 HRH3 (0.79) HRH3LOXL2ABATF10F11
SCHEMBL1459020 0.64 HRH3 (0.52) HRH3LOXL2ABATF10F11
SCHEMBL22990410 0.64 HRH3 (0.52) HRH3LOXL2ABATF10F11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006067462-A1 1,6 - SUBSTITUTED (3R,6R) -3- (2,3-DIHYDRO-1H-INDEN-2-YL)-2,5-PIPERAZINEDIONE DERIVATIVES AS OXYTOCIN RECEPTOR ANTAGONISTS FOR THE TREATMENT OF PRE-TERM LABOUR, DYSMENORRHEA AND ENDOMETRIOSIS GLAXO GROUP LIMITED (GB) 2006-06-29 WO disclosed