SCHEMBL8265136

SCHEMBL8265136

C[C@]1(CC2CCCC2)NC(=N)N(Cc2ccc(CN)cc2)C1=O

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 5/20 0.38
ALDH1A1 P00352 7/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
LMNA P02545 3/20 0.34
MAPK1 P28482 1/20 0.34
OPRL1 P41146 2/20 0.34
OPRM1 P35372 1/20 0.33
OPRK1 P41145 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.32
MTOR P42345 1/20 0.32
NPC1 O15118 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32
ELANE P08246 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14105052 0.99 BACE1 (0.39) BACE1ALDH1A1SMN1; SMN2LMNAMAPK1
SCHEMBL10305479 0.88 BACE1 (0.41) BACE1ALDH1A1SMN1; SMN2LMNAMAPK1
SCHEMBL8265240 0.80 BACE1 (0.43) BACE1ALDH1A1SMN1; SMN2LMNAMAPK1
SCHEMBL17550893 0.80 BACE1 (0.44) BACE1ALDH1A1SMN1; SMN2LMNANPC1
SCHEMBL7600289 0.80 BACE1 (0.46) BACE1NPC1RAB9A
SCHEMBL14643202 0.79 BACE1 (0.44) BACE1SMN1; SMN2LMNAKMT2AMTOR
SCHEMBL8265686 0.79 BACE1 (0.61) BACE1ALDH1A1SMN1; SMN2LMNAMAPK1
SCHEMBL7518723 0.79 BACE1 (0.45) BACE1SMN1; SMN2NPC1RAB9A
SCHEMBL7516202 0.79 BACE1 (0.63) BACE1
SCHEMBL14644350 0.79 BACE1 (0.46) BACE1SMN1; SMN2LMNAMTORNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1838304-B1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS SCHERING CORP (US) 2009-08-19 EP disclosed
WO-2008103351-A2 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS SCHERING CORPORATION (US) 2008-08-28 WO disclosed
WO-2006065277-A2 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS SCHERING CORPORATION (US) 2006-06-22 WO disclosed