SCHEMBL8267016

SCHEMBL8267016

C=CC[C@H]1C(=O)N(C)C(=N)N[C@]1(C)c1cc(-c2cccc(N)c2)cs1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 13/20 0.36
BRD4 O60885 1/20 0.31
CYP3A4 P08684 3/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
CYP2D6 P10635 2/20 0.31
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14106178 0.89 BACE1 (0.36) BACE1BRD4CYP3A4BACE2CYP2D6
SCHEMBL14105370 0.88 BACE1 (0.33) BACE1BRD4
SCHEMBL14105515 0.87 BACE1 (0.35) BACE1BRD4CYP3A4BACE2CYP2D6
SCHEMBL7539867 0.87 BACE1 (0.48) BACE1CYP3A4CYP2D6CYP2C9
SCHEMBL13407619 0.87 BACE1 (0.48) BACE1CYP3A4CYP2D6CYP2C9
SCHEMBL14105517 0.86 BACE1 (0.35) BACE1BRD4CYP3A4BACE2CYP2D6
SCHEMBL14106047 0.85 BACE1 (0.33) BACE1BACE2
SCHEMBL14105255 0.85 BACE1 (0.31) BACE1
SCHEMBL13558821 0.85 PIM1 (0.35) BACE1BACE2
SCHEMBL7536016 0.85 PIM1 (0.35) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006065277-A2 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS SCHERING CORPORATION (US) 2006-06-22 WO disclosed