SCHEMBL8269474

SCHEMBL8269474

CC1=NN(c2cccc(F)c2)C(N2CCN(c3nc(-c4ccncc4F)cc(=O)n3C)CC2)C1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 19/20 0.49
CYP2D6 P10635 6/20 0.49
CYP1A2 P05177 5/20 0.49
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL87858 0.79 GSK3B (0.51) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL8268075 0.74 GSK3B (0.63) GSK3BCYP2D6CYP1A2
SCHEMBL2116043 0.74 GSK3B (0.64) GSK3BCYP2D6CYP1A2
SCHEMBL87832 0.74 GSK3B (0.62) GSK3BCYP2D6CYP1A2
SCHEMBL88129 0.73 GSK3B (0.55) GSK3BCYP2D6CYP1A2CYP3A4
SCHEMBL88127 0.73 GSK3B (0.51) GSK3BCYP2D6CYP1A2
SCHEMBL87782 0.73 GSK3B (0.54) GSK3BCYP2D6CYP1A2
SCHEMBL81961 0.73 GSK3B (0.69) GSK3BCYP2D6CYP1A2
SCHEMBL87939 0.73 GSK3B (0.72) GSK3BCYP2D6CYP1A2
SCHEMBL695999 0.71 GSK3B (0.74) GSK3BCYP2D6CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006036015-A2 6- (PYRIDINYL) -4-PYRIMIDONE DERIVATES AS TAU PROTEIN KINASE 1 INHIBITORS MITSUBISHI PHARMA CORPORATION (JP) 2006-04-06 WO disclosed