SCHEMBL8273239

SCHEMBL8273239

CC#CCn1c(N(C)CC(C)N)nc2c1c(=O)n(Cc1cc3ccccc3c(N)n1)c(=O)n2C

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 0.43
CHRM1 P11229 2/20 0.43
FAP Q12884 6/20 0.42
POU2F2 P09086 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
POU2F1 P14859 1/20 0.39
CHRM3 P20309 1/20 0.39
HRH2 P25021 1/20 0.39
MC4R P32245 1/20 0.39
DPP8 Q6V1X1 1/20 0.39
DPP9 Q86TI2 1/20 0.39
GHSR Q92847 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13936235 0.91 DPP4 (0.42) DPP4CHRM1FAPPOU2F2ADORA3
SCHEMBL682159 0.87 DPP4 (0.45) DPP4CHRM1FAPPOU2F2ADORA3
SCHEMBL8272340 0.86 DPP4 (0.51) DPP4CHRM1FAPPOU2F2ADORA3
SCHEMBL4471876 0.86 DPP4 (0.58) DPP4CHRM1FAPPOU2F2ADORA3
SCHEMBL4471886 0.86 DPP4 (0.58) DPP4CHRM1FAPPOU2F2ADORA3
SCHEMBL4475662 0.86 DPP4 (0.58) DPP4CHRM1FAPPOU2F2ADORA3
SCHEMBL8272356 0.85 DPP4 (0.56) DPP4
SCHEMBL8272341 0.85 DPP4 (0.46) DPP4CHRM1FAPPOU2F2ADORA3
SCHEMBL13936215 0.85 DPP4 (0.59) DPP4CHRM1FAPPOU2F2ADORA3
SCHEMBL8273225 0.84 DPP4 (0.43) DPP4CHRM1FAPPOU2F2ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797093-B1 NOVEL 3-METHYL-7-BUTINYL-XANTHINES, PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM INT (DE) 2012-05-30 EP disclosed
WO-2006029769-A1 NOVEL 3-METHYL-7-BUTINYL-XANTHINES, PRODUCTION THEREOF, AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2006-03-23 WO disclosed