SCHEMBL8282185

SCHEMBL8282185

Cc1ccc(NC(=O)c2ccc(Cl)cc2)cc1Nc1nccc(-c2cccnc2)n1.O=C(Cl)c1ccc(Cl)cc1

nearest known ligand 0.93

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 13/20 0.93
ABL1 P00519 11/20 0.93
BCR P11274 8/20 0.93
PDGFRB P09619 5/20 0.93
EGFR P00533 1/20 0.79
PRKCA P17252 1/20 0.79
KIT P10721 7/20 0.77
KDR P35968 1/20 0.70
ABL2 P42684 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9677 0.96 PDGFRA (1.00) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL1656154 0.91 PDGFRA (0.90) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL3219611 0.90 PDGFRA (0.83) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL11932096 0.89 PDGFRA (0.86) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL9820 0.89 PDGFRA (1.00) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL3055349 0.88 PDGFRA (0.89) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL13498211 0.88 PDGFRA (0.88) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL9782 0.88 PDGFRA (1.00) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL29498750 0.88 PDGFRA (1.00) PDGFRAABL1BCRPDGFRBEGFR
SCHEMBL11927842 0.88 ABL1 (1.00) PDGFRAABL1BCRPDGFRBEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0564409-B1 Pyrimidin derivatives and process for their preparation NOVARTIS AG (CH) 2000-01-19 EP disclosed
EP-0564409-A1 Pyrimidin derivatives and process for their preparation CIBA-GEIGY AG (CH) 1993-10-06 EP disclosed