SCHEMBL8283277

SCHEMBL8283277

C=C1CCC(NC[C@@H](O)CCc2cc(F)cc(F)c2)(c2cccc(C(C)(C)C)c2)CC1

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 19/20 0.56
CTSD P07339 19/20 0.56
CYP3A4 P08684 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8283712 0.91 BACE1 (0.67) BACE1CTSDCYP3A4
SCHEMBL2876001 0.91 BACE1 (0.67) BACE1CTSDCYP3A4
SCHEMBL4263894 0.90 BACE1 (0.55) BACE1CTSDCYP3A4
SCHEMBL2876938 0.89 BACE1 (0.65) BACE1CTSD
SCHEMBL2873582 0.89 BACE1 (0.59) BACE1CTSDCYP3A4
SCHEMBL8283430 0.87 BACE1 (0.57) BACE1CTSD
SCHEMBL2870684 0.87 BACE1 (0.57) BACE1CTSD
SCHEMBL8282820 0.86 BACE1 (0.56) BACE1CTSDCYP3A4
SCHEMBL8283045 0.86 BACE1 (0.56) BACE1CTSD
SCHEMBL2874644 0.86 BACE1 (0.56) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005087215-A1 SUBSTITUTED UREA AND CARBAMATE, PHENACYL-2-HYDROXY-3-DIAMINOALKANE, AND BENZAMIDE-2-HYDROXY-3-DIAMINOALKANE ASPARTYL-PROTEASE INHIBITORS ELAN PHARMACEUTICALS, INC. (US) 2005-09-22 WO disclosed