SCHEMBL8286071

SCHEMBL8286071

CCCN(CCC)C(=O)c1cc(-c2nnc([C@@](C)(N)Cc3ccccc3)o2)cc(-c2ccccc2C#N)c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 7/20 0.49
BACE2 Q9Y5Z0 2/20 0.43
OXTR P30559 2/20 0.37
AVPR1A P37288 2/20 0.37
ALDH1A1 P00352 1/20 0.37
POLB P06746 1/20 0.37
CTSA P10619 1/20 0.36
APLNR P35414 1/20 0.34
CTSD P07339 5/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
KCNH2 Q12809 1/20 0.34
THRB P10828 1/20 0.33
MYC P01106 1/20 0.32
WDR5 P61964 1/20 0.32
FAAH O00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12993835 1.00 BACE1 (0.49) BACE1BACE2OXTRAVPR1AALDH1A1
SCHEMBL12993778 0.94 BACE1 (0.51) BACE1BACE2OXTRAVPR1AALDH1A1
SCHEMBL8284272 0.93 BACE1 (0.50) BACE1BACE2OXTRAVPR1AALDH1A1
SCHEMBL3592515 0.88 BACE1 (0.47) BACE1BACE2ALDH1A1POLBAPLNR
SCHEMBL8284287 0.88 BACE1 (0.47) BACE1BACE2ALDH1A1POLBAPLNR
SCHEMBL3592518 0.88 BACE1 (0.47) BACE1BACE2ALDH1A1POLBAPLNR
SCHEMBL3595507 0.88 BACE1 (0.52) BACE1BACE2ALDH1A1CTSAAPLNR
SCHEMBL3598706 0.88 BACE1 (0.52) BACE1BACE2ALDH1A1CTSAAPLNR
SCHEMBL3598702 0.88 BACE1 (0.52) BACE1BACE2ALDH1A1CTSAAPLNR
SCHEMBL12993809 0.88 BACE1 (0.51) BACE1BACE2OXTRAVPR1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005103020-A1 1,3,5-SUBSTITUTED PHENYL DERIVATIVE COMPOUNDS USEFUL AS BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE MERCK & CO., INC. (US) 2005-11-03 WO disclosed