SCHEMBL8286754

SCHEMBL8286754

COc1cccc(C(=O)N[C@H](C(=O)N2CCC[C@H]2C(=O)NCC=O)C(C)C)c1C

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.45
XIAP P98170 1/20 0.44
MLX Q9UH92 1/20 0.44
ELANE P08246 8/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TACR1 P25103 1/20 0.40
CTSG P08311 1/20 0.40
ATM Q13315 1/20 0.40
CCR1 P32246 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12949921 0.88 TAAR1 (0.54) TAAR1XIAPMLXELANECTSG
SCHEMBL3174391 0.86 KMT2A (0.49) ELANEMEN1KMT2ACCR1
SCHEMBL8288957 0.86 CCR1 (0.44) CCR1
SCHEMBL12747910 0.85 ELANE (0.46) XIAPMLXELANECTSG
SCHEMBL12949899 0.84 ELANE (0.48) TAAR1XIAPMLXELANECTSG
SCHEMBL12949783 0.83 TSHR (0.45) TAAR1XIAPMLXELANEMEN1
SCHEMBL12949915 0.83 TAAR1 (0.49) TAAR1XIAPMLXELANECTSG
SCHEMBL8287915 0.82 CCR1 (0.46) CCR1
SCHEMBL8286821 0.81 ELANE (0.43) ELANEMEN1KMT2ATACR1ATM
SCHEMBL12949987 0.81 TSHR (0.44) XIAPMLXMEN1KMT2ACCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005085236-A2 CASPASE INHIBITORS AND USES THEREOF VERTEX PHARMACEUTICALS INCORPORATED (US) 2005-09-15 WO disclosed