SCHEMBL8288298

SCHEMBL8288298

CCCCC1(c2cncc(-c3cccc(OC)c3)c2)NC(=N)C=C(C)CC1=O

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.36
CYP11B1 P15538 5/20 0.35
CYP11B2 P19099 5/20 0.35
BACE1 P56817 4/20 0.35
BACE2 Q9Y5Z0 1/20 0.35
KDR P35968 1/20 0.34
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
CYP1A2 P05177 2/20 0.33
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7524733 0.79 BACE1 (0.42) BRD4CYP11B1CYP11B2BACE1BACE2
SCHEMBL7580303 0.65 BACE1 (0.52) BRD4CYP11B1CYP11B2BACE1BACE2
SCHEMBL7524498 0.64 BACE1 (0.40) CYP11B1CYP11B2BACE1BACE2CYP3A4
SCHEMBL13557928 0.63 BACE1 (0.38) BRD4BACE1BACE2
SCHEMBL12108683 0.63 CYP11B1 (0.65) CYP11B1CYP11B2KDRCYP1A2CYP3A4
SCHEMBL7536107 0.62 BACE1 (0.54) CYP11B1CYP11B2BACE1BACE2CYP1A2
SCHEMBL11992511 0.61 CYP11B1 (0.54) CYP11B1CYP11B2CYP1A2CYP3A4CYP2C9
SCHEMBL7531592 0.59 BACE1 (0.53) BRD4BACE1BACE2
SCHEMBL14327635 0.59 CYP11B1 (0.52) CYP11B1CYP11B2BACE1CYP1A2CYP3A4
SCHEMBL14857157 0.59 BACE1 (0.47) BRD4CYP11B1CYP11B2BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005058311-A1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS SCHERING CORPORATION (US) 2005-06-30 WO disclosed