SCHEMBL8288369

SCHEMBL8288369

CCOC(=O)c1c(-c2ccc(Oc3ccccc3C#N)cc2)c(C#N)c(CC)n1C

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 19/20 0.60
GRIA4 P48058 19/20 0.60
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8287430 0.90 GRIA4 (0.74) GRIA2GRIA4
SCHEMBL4373075 0.90 GRIA2 (0.58) GRIA2GRIA4
SCHEMBL4373288 0.90 GRIA2 (0.55) GRIA2GRIA4
SCHEMBL8289329 0.89 GRIA4 (0.64) GRIA2GRIA4
SCHEMBL4537515 0.88 GRIA2 (0.59) GRIA2GRIA4
SCHEMBL4371248 0.86 GRIA2 (0.52) GRIA2GRIA4
SCHEMBL4374024 0.86 GRIA2 (0.77) GRIA2GRIA4
SCHEMBL13863270 0.86 GRIA2 (0.66) GRIA2GRIA4
SCHEMBL4373418 0.86 GRIA2 (0.56) GRIA2GRIA4
SCHEMBL8289332 0.85 GRIA2 (0.65) GRIA2GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1670757-B1 PYRROLE AND PYRAZOLE DERIVATIVES AS POTENTIATORS OF GLUTAMATE RECEPTORS LILLY CO ELI (US) 2009-05-06 EP disclosed
WO-2005040110-A1 PYRROLE AND PYRAZOLE DERIVATIVES AS POTENTIATORS OF GLUTAMATE RECEPTORS ELI LILLY AND COMPANY (US) 2005-05-06 WO disclosed