SCHEMBL8288495

SCHEMBL8288495

CSc1c(C#N)c(-c2ccc(-c3ccccc3C)cc2)c(C(=O)O)n1C

nearest known ligand 0.78

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GRIA4 P48058 20/20 0.78
GRIA2 P42262 18/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8288471 0.90 GRIA4 (0.80) GRIA4GRIA2
SCHEMBL4386187 0.89 GRIA4 (0.78) GRIA4GRIA2
SCHEMBL8289614 0.88 GRIA4 (1.00) GRIA4GRIA2
SCHEMBL8288359 0.86 GRIA4 (0.58) GRIA4GRIA2
SCHEMBL8289589 0.84 GRIA4 (0.72) GRIA4GRIA2
SCHEMBL8289467 0.84 GRIA4 (0.72) GRIA4GRIA2
SCHEMBL8289586 0.82 GRIA4 (0.79) GRIA4GRIA2
SCHEMBL13611802 0.82 GRIA4 (0.75) GRIA4GRIA2
SCHEMBL8287418 0.82 GRIA4 (1.00) GRIA4GRIA2
SCHEMBL8288484 0.80 GRIA4 (1.00) GRIA4GRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7625932-B2 Pyrrole and pyrazole derivatives as potentiators of glutamate receptors ELI LILLY AND COMPANY (US) 2009-12-01 US disclosed
EP-1670757-B1 PYRROLE AND PYRAZOLE DERIVATIVES AS POTENTIATORS OF GLUTAMATE RECEPTORS LILLY CO ELI (US) 2009-05-06 EP disclosed
US-20070066573-A1 Pyrrole and pyrazole derivatives as potentiators of glutamate receptors ELI LILLY AND COMPANY 2007-03-22 US disclosed
WO-2005040110-A1 PYRROLE AND PYRAZOLE DERIVATIVES AS POTENTIATORS OF GLUTAMATE RECEPTORS ELI LILLY AND COMPANY (US) 2005-05-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070066573-A1 Pyrrole and pyrazole derivatives as potentiators of glutamate receptors GRIN1, GRIN3A, GRIK5 GRIA4 16/4885GRIA2 17/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.