SCHEMBL8290353

SCHEMBL8290353

CCCCC1(CCCC)NC(=N)N(CC2CCN(C(=C3CC3)C(c3ccccc3)c3ccccc3)CC2)C1=O

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.33
OPRM1 P35372 2/20 0.32
OPRD1 P41143 2/20 0.32
OPRK1 P41145 2/20 0.32
OPRL1 P41146 2/20 0.32
CACNA2D1 P54289 1/20 0.31
CACNA1B Q00975 1/20 0.31
CACNB1 Q02641 1/20 0.31
CACNA1C Q13936 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7520707 0.88 TSHR (0.40) KMT2ACACNA2D1CACNA1BCACNB1CACNA1C
SCHEMBL7521187 0.81 CHRM3 (0.37) KMT2AALDH1A1LMNASMN1; SMN2
SCHEMBL7527644 0.79 POLB (0.46) KMT2AALDH1A1LMNASMN1; SMN2
SCHEMBL7522478 0.78 ATM (0.36) KMT2A
SCHEMBL7527772 0.78 KMT2A (0.44) KMT2AALDH1A1LMNASMN1; SMN2
SCHEMBL7525808 0.78 KMT2A (0.34) KMT2AALDH1A1LMNASMN1; SMN2
SCHEMBL7522795 0.77 KMT2A (0.42) KMT2A
SCHEMBL7529130 0.77 BACE1 (0.34) KMT2A
SCHEMBL7523899 0.77 IDH1 (0.35) KMT2ASMN1; SMN2
SCHEMBL13722775 0.77 GAA (0.42) KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005058311-A1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS SCHERING CORPORATION (US) 2005-06-30 WO disclosed