SCHEMBL8290653

SCHEMBL8290653

CC(=O)Nc1sc2c(c1C(N)=O)CCOC2

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 1/20 0.67
KDM4E B2RXH2 4/20 0.66
FLT3 P36888 3/20 0.66
MEN1 O00255 1/20 0.66
CYP1A2 P05177 1/20 0.66
CYP2C19 P33261 1/20 0.66
KMT2A Q03164 1/20 0.66
PTPRC P08575 1/20 0.58
PTPN2 P17706 1/20 0.58
PTPN1 P18031 1/20 0.58
PTPRB P23467 1/20 0.58
PTPRE P23469 1/20 0.58
CNR2 P34972 5/20 0.52
ALDH1A1 P00352 5/20 0.51
TSHR P16473 3/20 0.51
HPGD P15428 3/20 0.49
HSD17B10 Q99714 2/20 0.49
MAPK10 P53779 1/20 0.49
MDM2 Q00987 1/20 0.49
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5449075 0.89 CFTR (0.66) CFTRKDM4EFLT3MEN1CYP1A2
SCHEMBL5458508 0.87 CFTR (0.61) CFTRKDM4EFLT3MEN1CYP1A2
SCHEMBL5447630 0.87 CFTR (0.61) CFTRKDM4EFLT3MEN1CYP1A2
SCHEMBL5445117 0.86 PTPRC (0.65) CFTRKDM4EFLT3MEN1CYP1A2
SCHEMBL5455876 0.86 CFTR (0.60) CFTRKDM4EFLT3MEN1CYP1A2
SCHEMBL5455880 0.86 CFTR (0.60) CFTRKDM4EFLT3MEN1CYP1A2
SCHEMBL5453381 0.85 CFTR (0.66) CFTRKDM4EFLT3MEN1CYP1A2
SCHEMBL5445049 0.85 CFTR (0.60) CFTRKDM4EFLT3MEN1CYP1A2
SCHEMBL5467520 0.85 ANO1 (0.67) CFTRKDM4EFLT3MEN1CYP1A2
SCHEMBL5455685 0.85 CFTR (0.63) CFTRKDM4EFLT3MEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed