SCHEMBL8294384

SCHEMBL8294384

CCCN(CCC)C(=O)c1cc(C)cc(C(=O)N[C@@H](Cc2cc(F)cc(F)c2)[C@H](O)C2CN(Cc3ccccc3)CCN2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 1.00
CTSD P07339 2/20 0.76
CTSE P14091 2/20 0.76
BACE2 Q9Y5Z0 2/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13497500 1.00 BACE1 (1.00) BACE1CTSDCTSEBACE2
SCHEMBL12854878 1.00 BACE1 (1.00) BACE1CTSDCTSEBACE2
SCHEMBL8294383 0.90 BACE1 (0.82) BACE1
SCHEMBL13497585 0.89 BACE1 (1.00) BACE1CTSDCTSEBACE2
SCHEMBL13341065 0.89 BACE1 (1.00) BACE1CTSDCTSEBACE2
SCHEMBL12854864 0.89 BACE1 (1.00) BACE1CTSDCTSEBACE2
SCHEMBL12854872 0.88 BACE1 (0.81) BACE1CTSDCTSEBACE2
SCHEMBL13497537 0.88 BACE1 (0.81) BACE1CTSDCTSEBACE2
SCHEMBL13497441 0.88 BACE1 (1.00) BACE1
SCHEMBL8292705 0.88 BACE1 (1.00) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016876-A2 CYCLIC AMINE BACE-1 INHIBITORS HAVING A BENZAMIDE SUBSTITUENT SCHERING CORPORATION (US) 2005-02-24 WO disclosed