SCHEMBL8295484

SCHEMBL8295484

CO/N=C(/c1ccc(C)cc1)N(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
TDP1 Q9NUW8 1/20 0.41
SMN1; SMN2 Q16637 4/20 0.40
ALDH1A1 P00352 8/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.37
LMNA P02545 1/20 0.37
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
CYP1A2 P05177 1/20 0.37
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
HPGD P15428 2/20 0.35
GSK3B P49841 1/20 0.34
PKM P14618 1/20 0.33
HTT P42858 1/20 0.33
ATM Q13315 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
NLRP1 Q9C000 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18290561 0.77 MEN1 (0.49) MEN1KMT2ATDP1SMN1; SMN2ALDH1A1
SCHEMBL7862976 0.74 TDP1 (0.46) MEN1KMT2ATDP1SMN1; SMN2ALDH1A1
SCHEMBL12603677 0.72 CYP1A2 (0.51) KMT2ATDP1SMN1; SMN2ALDH1A1GAA
SCHEMBL6815200 0.72 CYP1A2 (0.51) KMT2ATDP1SMN1; SMN2ALDH1A1GAA
SCHEMBL16440164 0.72 CYP1A2 (0.51) KMT2ATDP1SMN1; SMN2ALDH1A1GAA
SCHEMBL13882951 0.71 SMN1; SMN2 (0.54) MEN1KMT2ASMN1; SMN2ALDH1A1MAPT
SCHEMBL14902858 0.71 SMN1; SMN2 (0.54) MEN1KMT2ASMN1; SMN2ALDH1A1MAPT
SCHEMBL25836970 0.71 MEN1 (0.44) MEN1KMT2ATDP1SMN1; SMN2ALDH1A1
SCHEMBL14176132 0.69 KMT2A (0.62) MEN1KMT2ASMN1; SMN2ALDH1A1LMNA
SCHEMBL13606731 0.68 SMN1; SMN2 (0.41) KMT2ATDP1SMN1; SMN2ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7250415-B2 1,1-Disubstitutedcycloalkyl-, glycinamidyl-, sulfonyl-amidino-, and tetrahydropyrimidinyl-containing diaminoalkyl, β-aminoacids, α-aminoacids and derivatives thereof as factor Xa inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-07-31 US disclosed
US-7250415-B2 1,1-Disubstitutedcycloalkyl-, glycinamidyl-, sulfonyl-amidino-, and tetrahydropyrimidinyl-containing diaminoalkyl, β-aminoacids, α-aminoacids and derivatives thereof as factor Xa inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-07-31 US disclosed
WO-2004108892-A2 1,1-DISUBSTITUTEDCYCLOALKYL-, GLYCINAMIDYL-, SULFONYL-AMIDINO-, AND TETRAHYDROPYRIMIDINYL-CONTAINING DIAMINOALKYL, β-AMINOACIDS, α-AMINOACIDS AND DERIVATIVES THEREOF AS FACTOR XA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-12-16 WO disclosed