SCHEMBL8296306

SCHEMBL8296306

CCOC(=O)Cc1c(C)[nH]c2ccc(Cl)cc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 1/20 0.55
PRSS2 P07478 1/20 0.55
PRSS3 P35030 1/20 0.55
KLK6 Q92876 1/20 0.55
SIRT1 Q96EB6 5/20 0.53
KDM4E B2RXH2 2/20 0.53
LMNA P02545 1/20 0.53
ADRA2A P08913 1/20 0.52
ADRA2B P18089 1/20 0.52
ADRA2C P18825 1/20 0.52
HTR7 P34969 1/20 0.52
HTR2B P41595 1/20 0.52
HTR6 P50406 1/20 0.52
ALDH1A1 P00352 3/20 0.51
MEN1 O00255 1/20 0.51
GAA P10253 1/20 0.51
MAPT P10636 1/20 0.51
KMT2A Q03164 1/20 0.51
HPGD P15428 2/20 0.50
TSPO P30536 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1757929 0.88 AKR1C2 (0.54) PRSS1PRSS2PRSS3KLK6SIRT1
SCHEMBL8291738 0.86 KDM4E (0.69) KLK6KDM4ELMNAALDH1A1MEN1
SCHEMBL6222629 0.85 GAA (0.63) KDM4ELMNAHTR7HTR6ALDH1A1
SCHEMBL10277244 0.84 KDM4E (0.51) KLK6KDM4ELMNAHTR7HTR6
SCHEMBL5190391 0.84 JAK2 (0.55) KDM4ELMNAALDH1A1MEN1GAA
SCHEMBL1191675 0.84 KDM4E (0.51) KLK6KDM4ELMNAALDH1A1MEN1
SCHEMBL11331437 0.83 KDM4E (0.49) PRSS1PRSS2PRSS3KLK6KDM4E
SCHEMBL8298998 0.83 KDM4E (0.51) PRSS1PRSS2PRSS3KLK6SIRT1
SCHEMBL1757962 0.83 KDM4E (0.73) PRSS1PRSS2PRSS3KLK6SIRT1
SCHEMBL7964334 0.83 HCRTR1 (0.69) KDM4ELMNAALDH1A1MEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620214-B1 1H-indole-3-acetic acid hydrazide sPLA2 inhibitors LILLY CO ELI (US) 1999-03-03 EP disclosed
US-5578634-A SEPTIC SHOCK TREATMENT ELI LILLY AND COMPANY (US) 1996-11-26 US disclosed
EP-0620214-A1 1H-indole-3-acetic acid hydrazide sPLA2 inhibitors ELI LILLY AND COMPANY (US) 1994-10-19 EP disclosed