SCHEMBL8297344

SCHEMBL8297344

C=C(CC)c1ccc(OC)c(OC)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
GAA P10253 2/20 0.59
TSHR P16473 3/20 0.55
CYP2C9 P11712 2/20 0.55
CYP2C19 P33261 2/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
PDE4A P27815 4/20 0.54
PDE4B Q07343 4/20 0.54
PDE4C Q08493 4/20 0.54
PDE4D Q08499 4/20 0.54
CA12 O43570 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
CA4 P22748 1/20 0.53
CA6 P23280 1/20 0.53
CA7 P43166 1/20 0.53
TPMT P51580 1/20 0.53
CA9 Q16790 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10131587 0.85 TSHR (0.52) MEN1KMT2AGAATSHRCYP2C9
SCHEMBL16795704 0.85 CYP2C9 (0.55) MEN1KMT2AGAATSHRCYP2C9
SCHEMBL8152340 0.83 CYP2C9 (0.53) MEN1KMT2AGAATSHRCYP2C9
SCHEMBL14611953 0.83 MAOB (0.58) MEN1KMT2AGAATSHRCYP2C9
SCHEMBL14375953 0.79 PDE4A (0.79) MEN1KMT2AGAATSHRCYP2C9
SCHEMBL7943556 0.78 CA12 (0.64) MEN1KMT2AGAATSHRCYP2C9
SCHEMBL18848298 0.78 CYP2C9 (0.61) MEN1KMT2AGAATSHRCYP2C9
SCHEMBL8296526 0.78 CYP2C9 (0.61) MEN1KMT2AGAATSHRCYP2C9
SCHEMBL14395698 0.78 CA12 (0.59) MEN1KMT2AGAATSHRCYP2C9
SCHEMBL9781940 0.77 MEN1 (0.59) MEN1KMT2AGAATSHRCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997836-A Inhibitor of platelet activating factor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed
EP-0368670-A1 Trisubstituted piperazine compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1990-05-16 EP disclosed