SCHEMBL8297635

SCHEMBL8297635

Bc1cnc2[nH]cc(C=O)c2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.51
CCNT1 O60563 1/20 0.38
CDK9 P50750 1/20 0.38
HASPIN Q8TF76 1/20 0.38
CYP2A6 P11509 2/20 0.37
IMPDH2 P12268 1/20 0.37
AXL P30530 2/20 0.36
ALDH1A1 P00352 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
TRIM24 O15164 1/20 0.33
TRIM33 Q9UPN9 1/20 0.33
PLG P00747 1/20 0.33
PLAU P00749 1/20 0.33
CDK8 P49336 1/20 0.32
TNIK Q9UKE5 1/20 0.32
BRD4 O60885 2/20 0.32
PIM3 Q86V86 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24764929 0.82 KMT2A (0.54) KMT2ACCNT1CDK9HASPINCYP2A6
SCHEMBL29950990 0.79 KMT2A (0.51) KMT2ACCNT1CDK9HASPINCYP2A6
SCHEMBL1713774 0.79 KMT2A (0.51) KMT2ACCNT1CDK9HASPINCYP2A6
SCHEMBL1713542 0.79 KMT2A (0.51) KMT2ACCNT1CDK9HASPINCYP2A6
SCHEMBL1337617 0.79 KMT2A (0.51) KMT2ACCNT1CDK9HASPINCYP2A6
SCHEMBL1563587 0.79 KMT2A (0.51) KMT2ACCNT1CDK9HASPINCYP2A6
SCHEMBL29953688 0.79 KMT2A (0.51) KMT2ACCNT1CDK9HASPINCYP2A6
SCHEMBL9906847 0.79 KMT2A (0.51) KMT2ACCNT1CDK9HASPINCYP2A6
SCHEMBL29953503 0.79 KMT2A (0.51) KMT2ACCNT1CDK9HASPINCYP2A6
SCHEMBL21902715 0.76 DYRK1A (0.38) AXLCDK8TNIKGSK3BMAP3K11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079133-A2 COMPOUNDS AND METHODS FOR KINASE MODULATION, AND INDICATIONS THEREFOR PLEXXIKON, INC. (US) 2011-06-30 WO disclosed
WO-2004101565-A2 JNK INHIBITORS EISAI CO., LTD. (JP) 2004-11-25 WO disclosed