SCHEMBL8301894

SCHEMBL8301894

C=C(O)C(C)(C)Cc1ccc(-c2cccc(-n3cc(C(=O)NC4CC4)c(=O)c4cccnc43)c2)cc1

nearest known ligand 0.88

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 16/20 0.88
PDE4B Q07343 15/20 0.88
PDE4C Q08493 15/20 0.88
PDE4D Q08499 15/20 0.88
KCNH2 Q12809 5/20 0.70
CYP2C9 P11712 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5934209 0.94 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DKCNH2
SCHEMBL5111855 0.90 PDE4A (0.83) PDE4APDE4BPDE4CPDE4DKCNH2
SCHEMBL5114088 0.89 PDE4A (0.83) PDE4APDE4BPDE4CPDE4DKCNH2
SCHEMBL5141241 0.88 PDE4A (0.90) PDE4APDE4BPDE4CPDE4DKCNH2
SCHEMBL5119683 0.88 PDE4A (0.86) PDE4APDE4BPDE4CPDE4DKCNH2
SCHEMBL8301920 0.88 PDE4A (0.81) PDE4APDE4BPDE4CPDE4DKCNH2
SCHEMBL5344071 0.86 KCNH2 (0.80) PDE4APDE4BPDE4CPDE4DKCNH2
SCHEMBL8300300 0.86 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DKCNH2
SCHEMBL5343986 0.86 KCNH2 (0.79) PDE4APDE4BPDE4CPDE4DKCNH2
SCHEMBL4790605 0.85 PDE4A (0.81) PDE4APDE4BPDE4CPDE4DKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004105698-A2 USE OF PHOSPHATASE INHIBITORS AS ADJUNCT THERAPY FOR PSYCHIATRIC DISORDERS MERCK & CO., INC. (US) 2004-12-09 WO disclosed
WO-2004048374-A1 4-OXO-1-(3-SUBSTITUTED PHENYL-1,4-DIHYDRO-1,8-NAPHTHYRIDINE-3-CARBOXAMIDE PHOSPHODIESTERASE-4 INHIBITORS MERCK FROSST CANADA & CO. (CA) 2004-06-10 WO disclosed