SCHEMBL8302086

SCHEMBL8302086

C=C(C)c1cc(CN2CCN(CCCCCC(c3ccc(F)cc3)c3ccc(F)cc3)CC2)cc(C(C)(C)C)c1O

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 12/20 0.82
ALDH1A1 P00352 4/20 0.45
TSHR P16473 3/20 0.45
GAA P10253 2/20 0.45
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.45
THRB P10828 1/20 0.45
HPGD P15428 1/20 0.45
MAPT P10636 3/20 0.45
KDM4E B2RXH2 2/20 0.45
HSD17B10 Q99714 1/20 0.42
HTR1A P08908 1/20 0.41
DRD2 P14416 1/20 0.41
DRD1 P21728 1/20 0.41
DRD4 P21917 1/20 0.41
DRD5 P21918 1/20 0.41
SLC6A2 P23975 1/20 0.41
HRH2 P25021 1/20 0.41
HTR1D P28221 1/20 0.41
HTR2A P28223 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5017474 0.91 KCNH2 (1.00) KCNH2ALDH1A1TSHRGAALMNA
SCHEMBL5024658 0.81 KCNH2 (1.00) KCNH2
SCHEMBL5026294 0.79 KCNH2 (1.00) KCNH2TSHRHTR1ADRD2DRD1
SCHEMBL5024699 0.77 KCNH2 (0.72) KCNH2TSHRHTR1ADRD2DRD1
SCHEMBL5024071 0.77 KCNH2 (0.82) KCNH2ALDH1A1GAAPOLBMAPT
SCHEMBL5080746 0.77 KCNH2 (0.81) KCNH2HTR1ADRD1DRD4DRD5
SCHEMBL5023974 0.76 KCNH2 (0.81) KCNH2TSHRLMNAHTR1ADRD2
SCHEMBL5023661 0.76 KCNH2 (0.75) KCNH2HTR1ADRD2DRD4DRD5
SCHEMBL5079870 0.76 KCNH2 (1.00) KCNH2TSHRHTR1ADRD2DRD1
SCHEMBL5023608 0.74 KCNH2 (0.81) KCNH2HTR1ADRD2DRD1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004089922-A2 CALCIUM CHANNEL INHIBITORS COMPRISING BENZHYDRIL SPACED FROM PIPERAZINE NEUROMED TECHNOLOGIES, INC. (CA) 2004-10-21 WO disclosed