SCHEMBL8302427

SCHEMBL8302427

COc1ccc(/C=C/c2c(Cl)cncc2Cl)c2c1OCCO2

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.41
LMNA P02545 4/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GAA P10253 2/20 0.34
NPC1 O15118 1/20 0.34
EGFR P00533 1/20 0.34
CYP1A1 P04798 4/20 0.33
CYP1A2 P05177 4/20 0.33
CYP1B1 Q16678 4/20 0.33
PDE4D Q08499 4/20 0.32
MAPT P10636 2/20 0.32
NFE2L2 Q16236 4/20 0.32
HTT P42858 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8302433 1.00 PDE4B (0.41) PDE4BLMNAALDH1A1KDM4EHSD17B10
SCHEMBL6837524 0.95 PDE4B (0.39) PDE4BLMNAALDH1A1KDM4EHSD17B10
SCHEMBL6837527 0.95 PDE4B (0.39) PDE4BLMNAALDH1A1KDM4EHSD17B10
SCHEMBL5723239 0.79 PDE4B (0.38) PDE4BALDH1A1KDM4EHSD17B10
SCHEMBL5722978 0.79 PDE4B (0.38) PDE4BGAANPC1CYP1A1CYP1A2
SCHEMBL5723244 0.79 PDE4B (0.38) PDE4BALDH1A1KDM4EHSD17B10
SCHEMBL5722989 0.79 PDE4B (0.38) PDE4BGAANPC1CYP1A1CYP1A2
SCHEMBL5723118 0.77 PDE4B (0.40) PDE4BALDH1A1CYP1A2PDE4D
SCHEMBL5723107 0.77 PDE4B (0.40) PDE4BALDH1A1CYP1A2PDE4D
SCHEMBL5723202 0.74 PDE4B (0.36) PDE4BPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0943613-A1 OXYGENIC HETEROCYCLIC COMPOUNDS KYOWA HAKKO KOGYO KABUSHIKI KAISHA (JP) 1999-09-22 EP disclosed