SCHEMBL8302624

SCHEMBL8302624

CNC1CCN(c2ccc(C(=O)OCc3ccccc3)cc2F)C1=O

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 1/20 0.47
SRD5A2 P31213 1/20 0.47
F10 P00742 7/20 0.43
LMNA P02545 3/20 0.42
MAPT P10636 3/20 0.42
BCHE P06276 2/20 0.42
RAB9A P51151 2/20 0.42
ALDH1A1 P00352 2/20 0.42
NPC1 O15118 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KMT2A Q03164 2/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
PRMT1 Q99873 1/20 0.39
HPGD P15428 2/20 0.39
TSHR P16473 1/20 0.39
JMJD6 Q6NYC1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14440621 0.90 SRD5A1 (0.45) SRD5A1SRD5A2F10LMNAMAPT
SCHEMBL8302634 0.86 SRD5A1 (0.43) SRD5A1SRD5A2F10ALDH1A1KMT2A
SCHEMBL4858641 0.86 SRD5A1 (0.43) SRD5A1SRD5A2F10ALDH1A1KMT2A
SCHEMBL5460656 0.85 SRD5A1 (0.47) SRD5A1SRD5A2LMNAMAPTBCHE
Hydrochloric Acid SCHEMBL5467892 0.84 SRD5A1 (0.46) SRD5A1SRD5A2LMNAMAPTBCHE
SCHEMBL5460647 0.79 F10 (0.68) F10
SCHEMBL5459034 0.78 F10 (0.73) F10
SCHEMBL5459037 0.78 F10 (0.73) F10
SCHEMBL5460632 0.77 F10 (0.60) F10
SCHEMBL8298647 0.76 F10 (0.54) F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004110434-A1 2-PYRROLIDONE DERIVATIVES AND USE THEREOF AS FACTOR XA INHIBITORS GLAXO GROUP LIMITED (GB) 2004-12-23 WO disclosed