SCHEMBL8305965

SCHEMBL8305965

CCc1ccc(CNC(=O)c2cc(=O)[nH]c3ccc(S(=O)(=O)N4CCCCCC4)cc23)cc1

nearest known ligand 0.82

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.82
MAPT P10636 3/20 0.67
TDP1 Q9NUW8 1/20 0.67
LMNA P02545 1/20 0.65
ALDH1A1 P00352 1/20 0.65
HTT P42858 1/20 0.65
RXFP1 Q9HBX9 1/20 0.65
BACE1 P56817 3/20 0.64
KDM4E B2RXH2 1/20 0.55
THRB P10828 1/20 0.55
POLB P06746 1/20 0.54
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312476 0.93 TP53 (0.79) TP53MAPTTDP1LMNAALDH1A1
SCHEMBL8312221 0.93 TP53 (0.79) TP53MAPTTDP1LMNAALDH1A1
SCHEMBL8312500 0.92 TP53 (0.78) TP53MAPTTDP1LMNAALDH1A1
SCHEMBL8311325 0.91 TP53 (0.77) TP53MAPTTDP1LMNAALDH1A1
SCHEMBL8312636 0.91 TP53 (0.77) TP53MAPTTDP1LMNAALDH1A1
SCHEMBL8311212 0.91 TP53 (0.76) TP53MAPTTDP1LMNAALDH1A1
SCHEMBL8311835 0.91 TP53 (0.76) TP53MAPTTDP1LMNAALDH1A1
SCHEMBL8306279 0.90 TP53 (0.75) TP53MAPTTDP1LMNAALDH1A1
SCHEMBL8308783 0.90 TP53 (0.75) TP53MAPTTDP1LMNAALDH1A1
SCHEMBL8312212 0.89 TP53 (0.82) TP53MAPTTDP1LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078731-A1 QUINOLINE-CARBOXYLIC ACIDS AND THE DERIVATIVES THEREOF, A FOCUSED LIBRARY 'CHEMICAL DIVERSITY RESEARCH INSTITUTE', LTD. (RU) 2004-09-16 WO disclosed