SCHEMBL8306211

SCHEMBL8306211

OCCOCCCCCCc1ccc(Cl)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
USP2 O75604 1/20 0.53
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.53
CYP3A4 P08684 1/20 0.53
MAPK1 P28482 1/20 0.53
CASP1 P29466 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
SLCO1B3 Q9NPD5 1/20 0.53
SLCO1B1 Q9Y6L6 1/20 0.53
KCNH2 Q12809 5/20 0.49
SLC6A2 P23975 2/20 0.49
HRH1 P35367 2/20 0.49
HRH3 Q9Y5N1 2/20 0.49
CHRM2 P08172 1/20 0.49
ADRA2C P18825 1/20 0.49
SLC6A4 P31645 1/20 0.49
SLC6A3 Q01959 1/20 0.49
CACNA1C Q13936 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6905786 0.91 KCNH2 (0.56) KCNH2SLC6A2HRH1HRH3CHRM2
SCHEMBL3169926 0.85 TAAR1 (0.45) MEN1KMT2AUSP2ALDH1A1LMNA
SCHEMBL9249000 0.82 SLC6A2 (0.64) MEN1KMT2AKCNH2SLC6A2HRH1
SCHEMBL9021231 0.82 KCNH2 (0.49) KCNH2SLC6A2HRH1HRH3CHRM2
SCHEMBL9154096 0.82 KCNH2 (0.49) KCNH2SLC6A2HRH1HRH3CHRM2
SCHEMBL9021167 0.82 KCNH2 (0.49) KCNH2SLC6A2HRH1HRH3CHRM2
SCHEMBL9021237 0.82 KCNH2 (0.49) KCNH2SLC6A2HRH1HRH3CHRM2
SCHEMBL9021947 0.82 KCNH2 (0.49) KCNH2SLC6A2HRH1HRH3CHRM2
SCHEMBL9021235 0.82 KCNH2 (0.49) KCNH2SLC6A2HRH1HRH3CHRM2
SCHEMBL9154394 0.82 KCNH2 (0.49) KCNH2SLC6A2HRH1HRH3CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915843-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSES SMITHKLINE BEECHAM PLC (GB) 1999-05-19 EP disclosed
WO-1997041098-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1997-11-06 WO disclosed