SCHEMBL8306619

SCHEMBL8306619

COCCNc1ccc2ncnc(Nc3ccc(OCc4ccccn4)c(C)c3)c2c1

nearest known ligand 0.72

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 14/20 0.72
ERBB2 P04626 10/20 0.72
LCK P06239 1/20 0.57
ALDH1A1 P00352 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48
TSHR P16473 2/20 0.48
CYP2C19 P33261 2/20 0.48
HSD17B10 Q99714 2/20 0.48
CLK4 Q9HAZ1 2/20 0.48
ALOX15 P16050 1/20 0.48
MAPK1 P28482 1/20 0.48
LMNA P02545 1/20 0.48
ERBB4 Q15303 2/20 0.47
ABCG2 Q9UNQ0 1/20 0.47
ERBB3 P21860 1/20 0.47
AURKA O14965 1/20 0.46
RPS6KB1 P23443 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8309603 0.90 EGFR (0.71) EGFRERBB2LCKERBB4ERBB3
SCHEMBL8307102 0.85 EGFR (0.76) EGFRERBB2LCKERBB4ABCG2
SCHEMBL4560407 0.85 EGFR (0.76) EGFRERBB2LCKCYP1A2CYP3A4
SCHEMBL8309272 0.85 EGFR (0.76) EGFRERBB2LCKLMNAERBB4
Hydrochloric Acid SCHEMBL6185804 0.84 EGFR (0.75) EGFRERBB2LCKCYP1A2CYP3A4
SCHEMBL8306859 0.84 EGFR (1.00) EGFRERBB2LCKERBB4ABCG2
SCHEMBL8309699 0.83 ERBB2 (0.68) EGFRERBB2LCKERBB4ERBB3
Hydrochloric Acid SCHEMBL8309362 0.83 EGFR (0.98) EGFRERBB2LCKERBB4ABCG2
SCHEMBL8308380 0.83 EGFR (0.82) EGFRERBB2LCKERBB4ABCG2
SCHEMBL8309178 0.82 EGFR (0.70) EGFRERBB2LCKERBB4AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0790986-B1 ANILINE DERIVATIVES ZENECA LTD (GB) 1999-01-20 EP disclosed
US-5821246-A USEFUL AS TYROSINE KINASE INHIBITORS AND FOR THE TREATMENT OF PROLIFERATIVE DISEASES SUCH AS CANCER ZENECA LIMITED (GB) 1998-10-13 US disclosed
EP-0790986-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1997-08-27 EP disclosed
WO-1996015118-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1996-05-23 WO disclosed