SCHEMBL8306746

SCHEMBL8306746

N#Cc1n[nH]cc1-c1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.42
LMNA P02545 3/20 0.42
METAP1 P53582 2/20 0.42
CCR1 P32246 2/20 0.42
CCR5 P51681 2/20 0.42
CCR8 P51685 2/20 0.42
CYP1A2 P05177 1/20 0.42
POLB P06746 1/20 0.42
BLM P54132 1/20 0.42
HIF1A Q16665 1/20 0.42
DOHH Q9BU89 1/20 0.42
P4HTM Q9NXG6 1/20 0.42
METAP2 P50579 2/20 0.39
NPC1 O15118 4/20 0.38
RAB9A P51151 4/20 0.38
GRM5 P41594 3/20 0.38
PRKCI P41743 1/20 0.37
TP53 P04637 3/20 0.37
TDP1 Q9NUW8 3/20 0.37
ALOX15 P16050 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17251975 0.75 KDM4E (0.48) KDM4ELMNAMETAP1CCR1CCR5
SCHEMBL1924499 0.75 KDM4E (0.48) KDM4ELMNAMETAP1CCR1CCR5
SCHEMBL31030262 0.75 KDM4E (0.48) KDM4ELMNAMETAP1CCR1CCR5
SCHEMBL3463943 0.75 KDM4E (0.48) KDM4ELMNAMETAP1CCR1CCR5
SCHEMBL11937882 0.75 ERBB2 (0.50) KDM4ECYP1A2METAP2GRM5ALOX15
SCHEMBL10921322 0.74 KDM4E (0.46) KDM4ELMNAMETAP1CCR1CCR5
SCHEMBL1384700 0.74 KDM4E (0.46) KDM4ELMNAMETAP1CCR1CCR5
SCHEMBL31339152 0.74 KDM4E (0.46) KDM4ELMNAMETAP1CCR1CCR5
SCHEMBL27917937 0.73 LRRK2 (0.42) KDM4ELMNAMETAP1CCR1CCR5
SCHEMBL8113038 0.72 SMN1; SMN2 (0.46) KDM4ELMNAMETAP1CCR1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024141444-A1 NEW BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2024-07-04 WO disclosed
WO-2023139085-A1 NEW BENZIMIDAZOLE PYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2023-07-27 WO disclosed
EP-0948487-A1 PESTICIDAL 1-ARYL AND PYRIDYLPYRAZOLE DERIVATIVES RHONE-POULENC AGROCHIMIE (FR) 1999-10-13 EP disclosed
WO-1998028279-A1 PESTICIDAL 1-ARYL AND PYRIDYLPYRAZOLE DERIVATIVES RHONE-POULENC AGROCHIMIE (FR) 1998-07-02 WO disclosed