SCHEMBL8306897

SCHEMBL8306897

NC(=O)C(N)c1cncnc1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.39
CYP19A1 P11511 2/20 0.33
LRRK2 Q5S007 1/20 0.33
CYP11B2 P19099 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
TSHR P16473 1/20 0.30
MC4R P32245 1/20 0.30
ADRA1A P35348 1/20 0.30
MC3R P41968 1/20 0.30
AR P10275 1/20 0.30
PLAU P00749 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25660370 0.82 HCAR2 (0.44) HCAR2
SCHEMBL1484347 0.76 EPHX1 (0.44) HCAR2CYP19A1LRRK2AR
SCHEMBL1354541 0.75 F7 (0.50) HCAR2
SCHEMBL1354543 0.75 F7 (0.50) HCAR2
SCHEMBL2178492 0.73 NAPRT (0.39) ADORA3
SCHEMBL2178495 0.73 NAPRT (0.39) ADORA3
SCHEMBL5399972 0.72 CYP2C9 (0.37) CYP11B2TSHR
SCHEMBL2438138 0.71 AKR1C3 (0.42) HCAR2AR
SCHEMBL28090653 0.69
SCHEMBL15797528 0.69 AKR1C3 (0.35) HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630244-B1 MUSCARINIC AGONISTS UNIV TOLEDO (US) 1999-12-01 EP disclosed
US-5403845-A Cognition activators; Alzheimer*s disaease UNIVERSITY OF TOLEDO (US) 1995-04-04 US disclosed
EP-0630244-A1 MUSCARINIC AGONISTS THE UNIVERSITY OF TOLEDO (US) 1994-12-28 EP disclosed
EP-0630244-A4 MUSCARINIC AGONISTS. UNIV TOLEDO (US) 1994-04-07 EP disclosed
WO-1993003726-A1 MUSCARINIC AGONISTS THE UNIVERSITY OF TOLEDO (US) 1993-03-04 WO disclosed
US-5175166-A Cognition activators THE UNIVERSITY OF TOLEDO (US) 1992-12-29 US disclosed