SCHEMBL8308611

SCHEMBL8308611

C/C(=N/OCCOc1ccc(CC2SC(=O)NC2=O)cc1)c1ccc(OCc2ccccc2)nc1

nearest known ligand 0.76

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PPARG P37231 12/20 0.76
FFAR1 O14842 9/20 0.52
PPARA Q07869 3/20 0.49
RXRA P19793 2/20 0.46
CYP3A4 P08684 1/20 0.46
RARG P13631 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8308613 1.00 PPARG (0.76) PPARGFFAR1PPARARXRACYP3A4
SCHEMBL6904420 0.90 PPARG (0.72) PPARGFFAR1PPARARXRACYP3A4
SCHEMBL6904419 0.90 PPARG (0.72) PPARGFFAR1PPARARXRACYP3A4
SCHEMBL6898686 0.89 PPARG (0.73) PPARGFFAR1PPARARXRACYP3A4
SCHEMBL6898681 0.89 PPARG (0.73) PPARGFFAR1PPARARXRACYP3A4
SCHEMBL6902809 0.87 PPARG (0.77) PPARGFFAR1RXRACYP3A4RARG
SCHEMBL6902815 0.87 PPARG (0.77) PPARGFFAR1RXRACYP3A4RARG
SCHEMBL6902220 0.86 PPARG (0.70) PPARGFFAR1PPARARXRACYP3A4
SCHEMBL6902217 0.86 PPARG (0.70) PPARGFFAR1PPARARXRACYP3A4
SCHEMBL6898697 0.86 PPARG (1.00) PPARGFFAR1RXRACYP3A4RARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5972959-A Oxime derivatives, their preparation and their therapeutic use SANKYO COMPANY, LIMITED (JP) 1999-10-26 US disclosed
EP-0708098-B1 Oxime derivatives, their preparation and their therapeutic use SANKYO CO (JP) 1999-03-03 EP disclosed
EP-0708098-A1 Oxime derivatives, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1996-04-24 EP disclosed