SCHEMBL8312606

SCHEMBL8312606

CCSc1cccc(Oc2ncc(F)cc2C(=O)NC2CCCCC2)c1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 17/20 0.51
PDE4A P27815 1/20 0.51
PDE4D Q08499 1/20 0.51
CNR2 P34972 2/20 0.46
HPGD P15428 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CNR1 P21554 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5839702 0.89 PDE4B (0.50) PDE4BPDE4APDE4D
SCHEMBL5839698 0.89 PDE4B (0.50) PDE4BPDE4APDE4D
SCHEMBL5839215 0.89 CNR1 (0.44) PDE4BPDE4APDE4DCNR1
SCHEMBL5840163 0.89 CNR1 (0.44) PDE4BPDE4APDE4DCNR1
SCHEMBL5778513 0.88 PTGER4 (0.43) PDE4BPDE4APDE4D
SCHEMBL5779293 0.87 PDE4B (0.49) PDE4BPDE4APDE4D
SCHEMBL5779289 0.87 PDE4B (0.49) PDE4BPDE4APDE4D
SCHEMBL5839350 0.87 PDE4B (0.49) PDE4BPDE4APDE4D
SCHEMBL5841960 0.83 PDE4B (0.53) PDE4BPDE4APDE4D
SCHEMBL5841951 0.83 PDE4B (0.53) PDE4BPDE4APDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005009966-A1 NICOTINAMIDE DERIVATIVES USEFUL AS PDE4 INHIBITORS PFIZER LIMITED (GB) 2005-02-03 WO disclosed