SCHEMBL8313136

SCHEMBL8313136

Cc1ncsc1-c1ccnc(Nc2ccc(Cl)nc2)n1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 18/20 0.52
CDK4 P11802 14/20 0.47
CDK1 P06493 4/20 0.47
CDK7 P50613 4/20 0.47
CDK9 P50750 4/20 0.47
AURKA O14965 3/20 0.47
AURKB Q96GD4 2/20 0.47
PLK1 P53350 3/20 0.46
CCNE1 P24864 3/20 0.45
CCNA2 P20248 1/20 0.44
CCNT1 O60563 1/20 0.43
CCNB1 P14635 1/20 0.43
CCND1 P24385 1/20 0.43
CCNH P51946 1/20 0.43
TNF P01375 1/20 0.41
SYK P43405 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314041 0.85 CDK2 (0.52) CDK2CDK4CDK1CDK7CDK9
SCHEMBL5620875 0.83 CDK2 (0.76) CDK2CDK4CDK1CDK7CDK9
SCHEMBL5785381 0.82 CDK2 (0.58) CDK2CDK4CDK1CDK7CDK9
SCHEMBL5620822 0.81 CDK2 (0.69) CDK2CDK4CDK1CDK7CDK9
SCHEMBL1415012 0.81 CDK2 (0.67) CDK2CDK4CDK1CDK7CDK9
SCHEMBL5621800 0.80 CDK2 (0.70) CDK2CDK4CDK1CDK7CDK9
SCHEMBL8311832 0.80 CLK4 (0.49) CDK2CDK4CDK1CDK7CDK9
SCHEMBL4397546 0.78 CDK2 (0.50) CDK2CDK4CDK1CDK7CDK9
SCHEMBL2087406 0.77 CDK2 (0.61) CDK2CDK4CDK1CDK7CDK9
SCHEMBL4388874 0.76 SYK (0.70) CDK2SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005012298-A1 PYRIDINYLAMINO-PYRIMIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS CYCLACEL LIMITED (GB) 2005-02-10 WO disclosed