SCHEMBL8313196

SCHEMBL8313196

CSc1cccc(Oc2ncc(F)cc2C(=O)N[C@H]2CC[C@@H](NC(=O)c3cccc4cc(O)cnc34)CC2)c1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 20/20 0.51
PDE4A P27815 1/20 0.51
PDE4D Q08499 1/20 0.51
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5855404 1.00 PDE4B (0.51) PDE4BPDE4APDE4DCYP3A4CYP2C9
SCHEMBL5856659 0.90 PDE4B (0.50) PDE4BPDE4APDE4D
SCHEMBL8313168 0.90 PDE4B (0.50) PDE4BPDE4APDE4D
SCHEMBL8312818 0.88 PDE4B (0.54) PDE4BPDE4APDE4DCYP3A4CYP2C9
SCHEMBL5840103 0.88 PDE4B (0.54) PDE4BPDE4APDE4DCYP3A4CYP2C9
SCHEMBL5750041 0.87 PDE4B (0.59) PDE4BPDE4APDE4DCYP3A4
SCHEMBL5840169 0.85 PDE4B (0.55) PDE4BPDE4APDE4DCYP3A4
SCHEMBL5780663 0.85 PDE4B (0.55) PDE4BPDE4APDE4DCYP3A4
SCHEMBL5840683 0.85 PDE4B (0.55) PDE4BPDE4APDE4DCYP3A4
SCHEMBL8313084 0.85 PDE4B (0.55) PDE4BPDE4APDE4DCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005010001-A1 NICOTINAMIDE DERIVATIVES USEFUL AS PDEA4 INHIBITORS PFIZER LIMITED (GB) 2005-02-03 WO disclosed