SCHEMBL8313754

SCHEMBL8313754

N#Cc1cc(Nc2ncnc3cnc(N[C@H]4CC[C@H](O)CC4)nc23)ccc1N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 6/20 0.51
EGFR P00533 6/20 0.49
ERBB2 P04626 1/20 0.49
HPGD P15428 1/20 0.49
HTT P42858 1/20 0.49
MAPK8 P45983 1/20 0.41
MAPK9 P45984 1/20 0.41
CHUK O15111 1/20 0.40
CDK1 P06493 1/20 0.40
GSK3A P49840 1/20 0.39
GSK3B P49841 1/20 0.39
FLT3 P36888 1/20 0.38
TYRO3 Q06418 1/20 0.38
MERTK Q12866 1/20 0.38
GAS6 Q14393 1/20 0.38
USP2 O75604 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8313760 1.00 BRAF (0.51) BRAFEGFRERBB2HPGDHTT
SCHEMBL6991635 0.89 EGFR (0.56) BRAFEGFRERBB2HPGDHTT
SCHEMBL8316968 0.89 EGFR (0.56) BRAFEGFRERBB2HPGDHTT
SCHEMBL6994918 0.87 EGFR (0.58) BRAFEGFRERBB2HPGDHTT
SCHEMBL6994924 0.87 EGFR (0.58) BRAFEGFRERBB2HPGDHTT
SCHEMBL6991028 0.82 GSK3A (0.55) BRAFEGFRERBB2HPGDHTT
SCHEMBL6991037 0.82 GSK3A (0.55) BRAFEGFRERBB2HPGDHTT
SCHEMBL8315344 0.81 EGFR (0.64) BRAFEGFRERBB2HPGDHTT
SCHEMBL8315620 0.81 EGFR (0.64) BRAFEGFRERBB2HPGDHTT
SCHEMBL8315348 0.81 EGFR (0.64) BRAFEGFRERBB2HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed